IDENTIFICATION OF BORTEZOMIB AS MYCOBACTERIAL CASEINOLYTIC PROTEASE INHIBITOR

IDENTIFICATION OF BORTEZOMIB AS MYCOBACTERIAL CASEINOLYTIC PROTEASE INHIBITOR

Ph.D

محفوظ في:

التفاصيل البيبلوغرافية
المؤلف الرئيسي:	GRACE NGAN JIE YIN
مؤلفون آخرون:	MICROBIOLOGY & IMMUNOLOGY
التنسيق:	Theses and Dissertations
اللغة:	English
منشور في:	2018
الموضوعات:	Bortezomib, Mycobacterium, Caseinolytic Protease, Inhibitor
الوصول للمادة أونلاين:	http://scholarbank.nus.edu.sg/handle/10635/144391
الوسوم:	إضافة وسم لا توجد وسوم, كن أول من يضع وسما على هذه التسجيلة!

مواد مشابهة

Functional studies of atypical caseinolytic protease subunits from Plasmodium falciparum
بواسطة: LIN WENJIE
منشور في: (2010)

Bortezomib warhead-switch confers dual activity against mycobacterial caseinolytic protease and proteasome and selectivity against human proteasome
بواسطة: Moreira W., وآخرون
منشور في: (2020)

IDENTIFICATION AND CHARACTERIZATION OF A PLASMODIUM VIVAX INHIBITOR OF CYSTEINE PROTEASES
بواسطة: LIM JUN JI
منشور في: (2014)

Structural Studies of Cysteine and Serine Protease Inhibitors Towards Therapeutic Applications
بواسطة: SHENOY RAJESH TULSIDAS
منشور في: (2011)

Synthesis of key intermediates towards HIV protease inhibitors
بواسطة: Prapapan Modhiran
منشور في: (2012)

Synthesis of key intermediates towards HIV protease inhibitors
بواسطة: Prapapan Modhiran
منشور في: (2007)

Mycobacterial caseinolytic protease gene regulator ClgR is a substrate of caseinolytic protease
بواسطة: Yamada Y., وآخرون
منشور في: (2020)

Target mechanism-based whole-cell screening identifies bortezomib as an inhibitor of caseinolytic protease in mycobacteria
بواسطة: Moreira W., وآخرون
منشور في: (2018)

A novel serine protease inhibitor acts as an immunomodulatory switch while maintaining homeostasis
بواسطة: Jiang, N., وآخرون
منشور في: (2014)

Zika virus protease : an antiviral drug target
بواسطة: Kang, CongBao, وآخرون
منشور في: (2020)

Protease inhibitor from chicken plasma : purification, characterization and its application in surimi
بواسطة: Saroat Rawdkuen
منشور في: (2005)

Towards selective mycobacterial ClpP1P2 inhibitors with reduced activity against the human proteasome
بواسطة: Moreira, W, وآخرون
منشور في: (2020)

Proteases from pyloric caeca of brownstripe red snapper (Lutjanus vitta): Purification, characterization and the use for production of hydrolysate with antioxidative activity
بواسطة: Sutheera Khantaphant
منشور في: (2011)

KAZAL TYPE PROTEASE INHIBITORS LEKTI AND KA69: STRUCTURE, FUNCTION AND IMPLICATION IN DISEASE
بواسطة: KARTHIK NAGAPPAN RAMESH
منشور في: (2017)

The impact of upfront versus sequential use of bortezomib among patients with newly diagnosed multiple myeloma (MM): A joint analysis of the Singapore MM Study Group and the Korean MM Working Party for the Asian myeloma network
بواسطة: Tan, D., وآخرون
منشور في: (2016)

Exploring the binding of peptidic West Nile virus NS2B-NS3 protease inhibitors by NMR
بواسطة: Kang, C., وآخرون
منشور في: (2014)

Attenuation of STAT3 signaling cascade by daidzin can enhance the apoptotic potential of bortezomib against multiple myeloma
بواسطة: Yang, M.H., وآخرون
منشور في: (2021)

Chemical biology of metalloproteases and cysteine proteases
بواسطة: HU MINGYU
منشور في: (2012)

Computational prediction of human immunodeficiency virus type 1 (HIV-1) protease inhibitors resistance using enzyme-ligand docking techniques
بواسطة: Ekachai Jenwitheesuk
منشور في: (2023)

Crystallization of a nonclassical Kazal-type Carcinoscorpius rotundicauda serine protease inhibitor, CrSPI-1, complexed with subtilisin
بواسطة: Tulsidas, S.R., وآخرون
منشور في: (2014)

Understanding the mechanism of action of protein synthesis inhibitors against Mycobacterium
بواسطة: LIM HAN WERN
منشور في: (2011)

Cloning and characterization of the alkaline protease gene (alpA) from Aspergillus oryzae
بواسطة: Supaporn Cheevadhanarak
منشور في: (2023)

Structure-guided fragment-based in silico drug design of dengue protease inhibitors
بواسطة: Knehans, T., وآخرون
منشور في: (2014)

Design, synthesis and biological evaluation of inhibitors of flavivirus NS2B/NS3 protease
بواسطة: GAO YAOJUN
منشور في: (2010)

Synthesis, evaluation and molecular modeling of chromone derivatives as HIV-1 protease inhibitors and molecular modeling of phthalimide derivatives as HIV-1 reverse transcriptase inhibitors
بواسطة: Weerasak Samee
منشور في: (2023)

Discovery, Synthesis, and invitro Evaluation of West Nile Virus Protease Inhibitors Based on the 9,10-Dihydro-3H,4aH-1,3,9,10a-tetraazaphenanthren-4-one Scaffold
بواسطة: Samanta, S., وآخرون
منشور في: (2014)

A male-specific (cysteine-rich) protein of Oesophagostomum dentatum (Strongylida) with structural characteristics of a serine protease inhibitor containing two trypsin inhibitor-like domains
بواسطة: Boag, P.R., وآخرون
منشور في: (2014)

Tripeptide inhibitors of dengue and West Nile virus NS2B-NS3 protease
بواسطة: Schüller, A., وآخرون
منشور في: (2014)

SYNTHESIS AND BIOLOGICAL EVALUATION OF SMALL MOLECULES AS INHIBITORS OF WEST NILE VIRUS NS2B-NS3 PROTEASE
بواسطة: SANJAY SAMANTA
منشور في: (2013)

Synthesis, anti HIV-1 protease activity and molecular modeling of non-peptidic chromone derivatives
بواسطة: Patcharawee Nunthanavanit
منشور في: (2023)

Synthesis and invitro Evaluation of West Nile Virus Protease Inhibitors Based on the 2-{6-[2-(5-Phenyl-4H-{1,2,4]triazol-3-ylsulfanyl)acetylamino]benzothiazol-2-ylsulfanyl}acetamide Scaffold
بواسطة: Samanta, S., وآخرون
منشور في: (2014)

Formononetin regulates multiple oncogenic signaling cascades and enhances sensitivity to bortezomib in a multiple myeloma mouse model
بواسطة: Kim, C., وآخرون
منشور في: (2021)

Dengue protease activity: The structural integrity and interaction of NS2B with NS3 protease and its potential as a drug target
بواسطة: Phong, W.Y., وآخرون
منشور في: (2014)

Structural basis for reversible and irreversible inhibition of human cathepsin L by their respective dipeptidyl glyoxal and diazomethylketone inhibitors
بواسطة: Shenoy, R.T., وآخرون
منشور في: (2014)

Recent developments in protease activity assays and sensors
بواسطة: Ong, I.L.H, وآخرون
منشور في: (2020)

Expedient solid-phase synthesis of both symmetric and asymmetric diol libraries targeting aspartic proteases
بواسطة: Shi, H., وآخرون
منشور في: (2014)

Effectiveness of Protease Inhibitor/Nucleos(t)ide Reverse Transcriptase Inhibitor-Based Second-line Antiretroviral Therapy for the Treatment of Human Immunodeficiency Virus Type 1 Infection in Sub-Saharan Africa: A Systematic Review and Meta-analysis
بواسطة: Stockdale A.J., وآخرون
منشور في: (2019)

Structure, dynamics and binding of drug resistance HIV-1 protease with major mutations
بواسطة: Ornjira Aruksakunwong
منشور في: (2011)

Structure, dynamics and binding of drug resistance HIV-1 protease with major mutations
بواسطة: Ornjira Aruksakunwong
منشور في: (2006)

Docking study of chromone derivatives as HIV-1 protease inhibitors
بواسطة: Jiraporn Ungwitayatorn, وآخرون
منشور في: (2010)